Lamivudine Triphosphate

Lamivudine Triphosphate

SCHEMBL2223243

Nc1ccn([C@H]2CS[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O2)c(=O)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLG P54098 3/20 1.00
CACNA1F O60840 2/20 0.62
LMNA P02545 2/20 0.62
ALB P02768 2/20 0.62
MAPT P10636 2/20 0.62
CACNA1D Q01668 2/20 0.62
CACNA1S Q13698 2/20 0.62
CACNA1C Q13936 2/20 0.62
PDE3A Q14432 2/20 0.62
POLB P06746 1/20 0.53
P2RY2 P41231 9/20 0.52
P2RY4 P51582 5/20 0.52
P2RY6 Q15077 4/20 0.52
P2RY12 Q9H244 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lamivudine Triphosphate SCHEMBL12595501 1.00 POLG (1.00) POLGCACNA1FLMNAALBMAPT
Lamivudine Triphosphate SCHEMBL14354589 1.00 POLG (1.00) POLGCACNA1FLMNAALBMAPT
SCHEMBL12595493 0.90 POLG (0.81) POLGCACNA1FLMNAALBMAPT
SCHEMBL30695575 0.90 POLG (0.81) POLGCACNA1FLMNAALBMAPT
SCHEMBL12595497 0.87 POLG (0.77) POLGCACNA1FLMNAALBMAPT
Emtricitabine 5'-Triphosphate SCHEMBL30480833 0.83 POLG (1.00) POLGCACNA1FLMNAALBMAPT
Emtricitabine 5'-Triphosphate SCHEMBL14354587 0.83 POLG (1.00) POLGCACNA1FLMNAALBMAPT
Emtricitabine 5'-Triphosphate SCHEMBL606449 0.83 POLG (1.00) POLGCACNA1FLMNAALBMAPT
Ddctp SCHEMBL18840498 0.82 POLG (0.70) POLGCACNA1FLMNAALBMAPT
Ddctp SCHEMBL16807754 0.82 POLG (0.70) POLGCACNA1FLMNAALBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2515908-A2 1,4-SUBSTITUTED PIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF Merck Sharp & Dohme Corp. (US) 2012-10-31 EP disclosed
WO-2011087738-A2 1,4-SUBSTITUTED PIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF SCHERING CORPORATION (US) 2011-07-21 WO disclosed
US-20030195239-A1 Inhibitors of hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same PFIZER INC. 2003-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030195239-A1 Inhibitors of hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same POLRMT, RNGTT, RNASE1 POLG 37/4885CACNA1F 4321/4885LMNA 3489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.