SCHEMBL2223717

SCHEMBL2223717

CCCN(C(=O)O)c1cccc(Cc2nn(-c3cc(F)cc(F)c3)ccc2=O)c1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
PDE10A Q9Y233 1/20 0.33
THRB P10828 1/20 0.32
LTB4R2 Q9NPC1 3/20 0.32
CACNA2D1 P54289 2/20 0.32
TP53 P04637 2/20 0.32
ACHE P22303 1/20 0.32
RAB9A P51151 2/20 0.31
NPC1 O15118 1/20 0.31
JAK2 O60674 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
PAX8 Q06710 1/20 0.31
KDM4E B2RXH2 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KAT6A Q92794 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
KLKB1 P03952 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2220259 0.92 TP53 (0.36) KMT2AMEN1PDE10ATP53RAB9A
SCHEMBL2223741 0.92 PDE10A (0.34) KMT2AMEN1PDE10ATHRBCACNA2D1
SCHEMBL2220196 0.91 ELOVL1 (0.37) THRBTP53
SCHEMBL13275659 0.90 KDM4E (0.34) KMT2AMEN1PDE10ACACNA2D1RAB9A
SCHEMBL2221341 0.90 PDE10A (0.33) KMT2AMEN1PDE10ACACNA2D1TP53
SCHEMBL2271255 0.90 PDE10A (0.33) KMT2AMEN1PDE10ALTB4R2CACNA2D1
SCHEMBL2221099 0.89 TP53 (0.38) KMT2AMEN1CACNA2D1TP53RAB9A
SCHEMBL13507151 0.88 KMT2A (0.33) KMT2AMEN1PDE10ACACNA2D1RAB9A
SCHEMBL13275023 0.87 KDM4E (0.32) KMT2AMEN1PDE10AKDM4EL3MBTL1
SCHEMBL2362163 0.87 OPRM1 (0.36) CACNA2D1ACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed