SCHEMBL2220196

SCHEMBL2220196

CCCN(C(=O)O)c1cccc(Cc2nn(-c3cncc(F)c3)ccc2=O)c1

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ELOVL1 Q9BW60 14/20 0.37
TP53 P04637 2/20 0.35
GRM2 Q14416 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2222078 0.93 ELOVL1 (0.38) ELOVL1TP53
SCHEMBL2223717 0.91 KMT2A (0.33) TP53THRB
SCHEMBL2222006 0.88 GRM2 (0.40) TP53GRM2
SCHEMBL2221099 0.87 TP53 (0.38) TP53GRM2
SCHEMBL2223741 0.86 PDE10A (0.34) TP53THRB
SCHEMBL2221341 0.85 PDE10A (0.33) TP53
SCHEMBL2220259 0.83 TP53 (0.36) TP53
SCHEMBL2221804 0.83 ENPP2 (0.35) TP53GRM2
SCHEMBL2219994 0.83 MEN1 (0.37)
SCHEMBL13275659 0.81 KDM4E (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO claimed