SCHEMBL22239262

SCHEMBL22239262

Oc1ccc(CCCN2CC3CCCC3C2)nc1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.42
GRIN2B Q13224 14/20 0.38
GRIN1 Q05586 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22239258 0.92 HRH3 (0.41) HRH3GRIN2BGRIN1
SCHEMBL29036770 0.80 CYP2D6 (0.52) HRH3
SCHEMBL22239201 0.78 HRH3 (0.47) HRH3
SCHEMBL29036764 0.75 NOS3 (0.46) HRH3
SCHEMBL29036763 0.75 CYP2D6 (0.51) HRH3
SCHEMBL24136402 0.74 GRIN2B (0.39) GRIN2BGRIN1
SCHEMBL29036801 0.74 HRH3 (0.49) HRH3
SCHEMBL22239303 0.72 GRIN2B (0.67) GRIN2BGRIN1
SCHEMBL24136364 0.72 GRIN2B (0.67) GRIN2BGRIN1
SCHEMBL29346469 0.72 GRIN2B (0.67) GRIN2BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3683207-A1 N-ALKYLARYL-5-OXYARYL-OCTAHYDRO-CYCLOPENTA[C]PYRROLE NEGATIVE ALLOSTERIC MODULATORS OF NR2B Cadent Therapeutics, Inc. (US) 2020-07-22 EP disclosed