SCHEMBL22239269

SCHEMBL22239269

Cc1ccc(C(=O)CN2CC3CCC[C@@]3(N)C2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.46
MEN1 O00255 4/20 0.46
ALDH1A1 P00352 6/20 0.44
GRIN2B Q13224 5/20 0.42
CYP1A1 P04798 2/20 0.38
CYP1B1 Q16678 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26020473 0.89 GRIN2B (0.47) GRIN2B
SCHEMBL24136445 0.75 GRIN2B (0.50) GRIN2B
SCHEMBL22239252 0.75 GRIN2B (0.40) GRIN2B
SCHEMBL17643340 0.74 GRIN2B (0.47) GRIN2B
SCHEMBL24136404 0.73 GRIN2B (0.37) GRIN2B
SCHEMBL24270959 0.72 MEN1 (0.56) KMT2AMEN1ALDH1A1GRIN2BSMN1; SMN2
SCHEMBL26021378 0.70 GRIN2B (0.36) GRIN2BMAPK1
SCHEMBL24271004 0.69
SCHEMBL4936082 0.69 MEN1 (0.75) KMT2AMEN1ALDH1A1CYP1A1CYP1B1
SCHEMBL6397229 0.68 KMT2A (0.59) KMT2AMEN1ALDH1A1GRIN2BMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3683207-A1 N-ALKYLARYL-5-OXYARYL-OCTAHYDRO-CYCLOPENTA[C]PYRROLE NEGATIVE ALLOSTERIC MODULATORS OF NR2B Cadent Therapeutics, Inc. (US) 2020-07-22 EP disclosed