SCHEMBL22239476

SCHEMBL22239476

CC(N)(O)CN1CNc2ccc(-c3cccc(C(F)(F)F)c3)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.38
KDM1A O60341 1/20 0.38
KIF11 P52732 1/20 0.37
PARP10 Q53GL7 1/20 0.37
PARP11 Q9NR21 1/20 0.37
S1PR5 Q9H228 1/20 0.36
SLC13A5 Q86YT5 1/20 0.36
IKBKB O14920 1/20 0.36
ASIC3 Q9UHC3 1/20 0.36
SLC6A7 Q99884 1/20 0.35
PIM1 P11309 1/20 0.35
BACE1 P56817 1/20 0.34
SLC1A3 P43003 2/20 0.34
SLC1A2 P43004 2/20 0.34
SLC1A1 P43005 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
SPHK2 Q9NRA0 1/20 0.34
SPHK1 Q9NYA1 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20393281 0.91 PARP10 (0.38) MAOBKDM1AKIF11PARP10PARP11
SCHEMBL18638653 0.82 PARP10 (0.38) MAOBKDM1AKIF11PARP10PARP11
SCHEMBL18638540 0.80 KIF11 (0.39) KIF11HRH3
SCHEMBL20393147 0.76 APP (0.42)
SCHEMBL18638342 0.71 KIF11 (0.36) KIF11HRH3
SCHEMBL18638629 0.69 PGR (0.38)
SCHEMBL11347344 0.69 MAPT (0.45) KIF11HRH3
SCHEMBL18638328 0.68 PIK3CD (0.32)
SCHEMBL18638664 0.67 APP (0.42)
SCHEMBL18638568 0.66 FGFR1 (0.32) PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3348547-B1 BENZIMIDAZOLE DERIVATIVES AS NAV 1.7 (SODIUM CHANNEL, VOLTAGE-GATED, TYPE IX, ALPHA SUBUNIT (SCN9A)) INHIBITORS FOR TREATING PAIN, DYSURIA AND MULTIPLE SCLEROSIS SUMITOMO DAINIPPON PHARMA CO LTD (JP) 2020-07-22 EP disclosed