SCHEMBL22239486

SCHEMBL22239486

O=CN1CCCC(c2cc(Cl)nc(C3CCOC3)n2)C1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAP3K12 Q12852 4/20 0.41
UCHL1 P09936 1/20 0.32
PIK3CA P42336 1/20 0.30
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22239462 0.79 PDE4B (0.33) MAP3K12
SCHEMBL16220399 0.77 TRPV3 (0.41) MAP3K12
SCHEMBL31568039 0.68 GSK3A (0.39)
SCHEMBL16220100 0.65 CNR2 (0.32)
SCHEMBL1616409 0.65 MAPT (0.43) MAP3K12PIK3CA
SCHEMBL855517 0.65 PIK3CA (0.38) PIK3CAMTOR
SCHEMBL23073961 0.64 HSD11B1 (0.39)
SCHEMBL13592662 0.64 HSD11B1 (0.39)
SCHEMBL16212243 0.64 MAP3K12 (0.37) MAP3K12
SCHEMBL19894137 0.63 PDE10A (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991977-B1 C-LINKED HETEROCYCLOALKYL SUBSTITUTED PYRIMIDINES AND THEIR USES HOFFMANN LA ROCHE (CH) 2020-07-22 EP disclosed