SCHEMBL22246232

SCHEMBL22246232

Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3P(C)C)n2)ccc1N1CCC2(CC1)CC(N)C2

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK9 P45984 3/20 0.55
MAPK10 P53779 3/20 0.55
EGFR P00533 7/20 0.54
ALK Q9UM73 3/20 0.47
CCNA2 P20248 5/20 0.47
CDK2 P24941 5/20 0.47
CCNK O75909 4/20 0.46
CCND3 P30281 4/20 0.46
CDK9 P50750 4/20 0.46
CDK6 Q00534 4/20 0.46
TNK2 Q07912 1/20 0.45
MAPK8 P45983 1/20 0.44
SRC P12931 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22246276 0.94 EGFR (0.49) MAPK9MAPK10EGFRALKCCNA2
SCHEMBL30503703 0.92 MAPK9 (0.55) MAPK9MAPK10EGFRALKCCNA2
SCHEMBL30503705 0.92 MAPK9 (0.53) MAPK9MAPK10EGFRCCNA2CDK2
SCHEMBL22246278 0.90 ALK (0.45) MAPK9MAPK10EGFRALKMAPK8
SCHEMBL22246265 0.89 EGFR (0.53) MAPK9MAPK10EGFRALKCCNA2
SCHEMBL22246172 0.89 MAPK9 (0.54) MAPK9MAPK10EGFRALKCCNA2
SCHEMBL30503727 0.88 MAPK9 (0.57) MAPK9MAPK10EGFRALKCCNA2
SCHEMBL30948591 0.88 MAPK9 (0.44) MAPK9MAPK10EGFRALKMAPK8
SCHEMBL30503717 0.88 MAPK9 (0.51) MAPK9MAPK10EGFRALKCCNA2
SCHEMBL30503700 0.87 EGFR (0.48) MAPK9MAPK10EGFRALKCCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113302196-B EGFR inhibitor, composition and application thereof 贝达药业股份有限公司 2023-08-04 CN disclosed
WO-2020147702-A1 EGFR INHIBITORS, COMPOSITIONS AND METHODS THEREOF BETTA PHARMACEUTICALS CO., LTD (CN) 2020-07-23 WO disclosed