SCHEMBL22248694

SCHEMBL22248694

Nc1ccn(-c2ccc(CN3CC4CCC(C3)C4N)cc2)c(=O)n1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.49
BTK Q06187 2/20 0.35
LIPE Q05469 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
MCHR1 Q99705 2/20 0.33
DPP4 P27487 2/20 0.32
DPP8 Q6V1X1 2/20 0.32
GRIN2B Q13224 1/20 0.32
KCNH2 Q12809 1/20 0.31
JAK1 P23458 1/20 0.31
JAK3 P52333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22249164 0.88 ROCK2 (0.47) ROCK2BTKLIPEHRH3MCHR1
SCHEMBL22248938 0.88 ROCK2 (0.48) ROCK2HRH3MCHR1DPP4DPP8
SCHEMBL22249157 0.88 ROCK2 (0.48) ROCK2HRH3MCHR1DPP4DPP8
SCHEMBL22254490 0.88 ROCK2 (0.49) ROCK2HRH3MCHR1DPP4DPP8
SCHEMBL22248366 0.86 ROCK2 (0.49) ROCK2LIPEHRH3MCHR1
SCHEMBL22254826 0.85 ROCK2 (0.49) ROCK2BTKLIPEHRH3MCHR1
SCHEMBL22254520 0.83 ROCK2 (0.48) ROCK2HRH3MCHR1JAK1JAK3
SCHEMBL22248654 0.83 ROCK2 (0.50) ROCK2HRH3
SCHEMBL22249176 0.83 ROCK2 (0.47) ROCK2BTKLIPEHRH3MCHR1
SCHEMBL22248937 0.82 ROCK2 (0.47) ROCK2HRH3MCHR1JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150372-A1 ANTIMICROBIAL COMPOUNDS AND METHODS CURZA GLOBAL, LLC (US) 2020-07-23 WO disclosed