SCHEMBL2225280

SCHEMBL2225280

CC(C)(C)C#Cc1cc(NC2CCC3(CC2)OCCO3)c(C(=O)O)s1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.39
NR1I2 O75469 2/20 0.36
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669322 0.90 ALDH1A1 (0.33) CYP2E1NR1I2RAB9ASMN1; SMN2ALDH1A1
SCHEMBL15015340 0.83 RAB9A (0.42) CYP2E1NR1I2RAB9ASMN1; SMN2L3MBTL1
SCHEMBL14647676 0.82 PIM1 (0.39) CYP2E1NR1I2RAB9ASMN1; SMN2
SCHEMBL12518971 0.81 NR1I2 (0.38) CYP2E1NR1I2RAB9ASMN1; SMN2L3MBTL1
SCHEMBL12518984 0.81 NR1I2 (0.38) CYP2E1NR1I2RAB9ASMN1; SMN2L3MBTL1
SCHEMBL15015264 0.80 CYP2E1 (0.42) CYP2E1NR1I2
SCHEMBL12949303 0.80 CYP2E1 (0.42) CYP2E1NR1I2
SCHEMBL12444669 0.79 RAF1 (0.34) CYP2E1NR1I2RAB9ASMN1; SMN2
SCHEMBL12444667 0.79 RAF1 (0.34) CYP2E1NR1I2RAB9ASMN1; SMN2
SCHEMBL2218006 0.79 RAF1 (0.34) CYP2E1NR1I2RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3219713-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES Gilead Sciences, Inc. (US) 2017-09-20 EP disclosed
EP-2523950-B1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES INC (US) 2017-03-15 EP disclosed
EP-2523950-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES Gilead Sciences, Inc. (US) 2012-11-21 EP disclosed
WO-2011088345-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES, INC. (US) 2011-07-21 WO disclosed