SCHEMBL22258595

SCHEMBL22258595

CCC(CC)C(=O)Nc1c[nH]nc1-c1nc2c([nH]1)CCN(C)C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 3/20 0.35
JAK3 P52333 3/20 0.35
JAK2 O60674 2/20 0.35
TYK2 P29597 2/20 0.35
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
POLB P06746 2/20 0.32
MAPK1 P28482 2/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TSHR P16473 2/20 0.32
GAA P10253 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
KDR P35968 1/20 0.31
LMNA P02545 1/20 0.31
KMT2A Q03164 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
FASN P49327 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22236261 0.81 ROCK2 (0.38) POLBMAPT
SCHEMBL5102502 0.78 HTR1F (0.43) JAK1JAK3JAK2TYK2HRH4
SCHEMBL5105549 0.78 HTR1F (0.39) JAK1JAK3JAK2TYK2KDM4E
SCHEMBL5112753 0.78 PDCD1 (0.39) JAK1JAK3JAK2TYK2POLB
SCHEMBL5111914 0.76 BRPF1 (0.44) KDM4EALDH1A1POLBMAPK1HSD17B10
SCHEMBL5103199 0.74 CYP2C19 (0.38) JAK1JAK3JAK2TYK2KDR
SCHEMBL5106436 0.74 ABL1 (0.43) ALDH1A1POLBGAAKMT2ACYP2C19
SCHEMBL22235779 0.72 GRIA1 (0.37) JAK1JAK3JAK2TYK2KDR
SCHEMBL5106326 0.70 HTR1F (0.40) JAK1JAK3KDM4EALDH1A1POLB
SCHEMBL5106208 0.68 ATR (0.38) POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020150545-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF THE WNT/B-CATENIN SIGNALING PATHWAY SAMUMED, LLC (US) 2020-07-23 WO disclosed