SCHEMBL22263187

SCHEMBL22263187

C=Cc1c(C(N)=O)cccc1-c1ccccc1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.53
PDK2 Q15119 1/20 0.42
SCN9A Q15858 5/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
BCAT2 O15382 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
CDC7 O00311 1/20 0.39
ROCK2 O75116 1/20 0.39
MAP4K4 O95819 1/20 0.39
PIM1 P11309 1/20 0.39
PRKACA P17612 1/20 0.39
CDK7 P50613 1/20 0.39
CDK9 P50750 1/20 0.39
HIPK2 Q9H2X6 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
SLC9A1 P19634 1/20 0.39
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30608075 0.81 PARP1 (0.56) PARP1PDK2SCN9ALMNAGAA
SCHEMBL5143960 0.81 PARP1 (0.56) PARP1PDK2SCN9ALMNAGAA
SCHEMBL22263186 0.81 PARP1 (0.48) PARP1PDK2SCN9ALMNAGAA
SCHEMBL4776527 0.79 PARP1 (0.54) PARP1PDK2SCN9ALMNAGAA
SCHEMBL29733181 0.79 PARP1 (0.58) PARP1PDK2SCN9ALMNAGAA
SCHEMBL6173688 0.78 PARP1 (0.53) PARP1PDK2SCN9ALMNAGAA
SCHEMBL3511705 0.76 PARP1 (0.47) PARP1LMNAGAABCAT2KEAP1
SCHEMBL2484725 0.75 PARP1 (0.49) PARP1PDK2SCN9ALMNAGAA
SCHEMBL26669294 0.74 PARP1 (0.50) PARP1PDK2SCN9ALMNAGAA
SCHEMBL2975349 0.74 PARP1 (0.39) PARP1GAAIRAK4ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11166460-B2 α-amino acrylate microbicide, and preparation method therefor and uses thereof NANKAI UNIVERSITY (CN) 2021-11-09 US disclosed
US-20200236935-A1 a-Amino Acrylate microbicide, and preparation method therefor and uses thereof UNIV NANKAI (CN) 2020-07-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200236935-A1 a-Amino Acrylate microbicide, and preparation method therefor and uses thereof AASDHPPT, ACE, ADA PARP1 1358/4885PDK2 3214/4885SCN9A 3224/4885
US-11166460-B2 α-amino acrylate microbicide, and preparation method therefor and uses thereof ACE, AASDHPPT, DDT PARP1 1364/4885PDK2 2801/4885SCN9A 2592/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.