SCHEMBL9980416

SCHEMBL9980416

CC1CCCN1c1ccc(S(N)(=O)=O)cc1CNc1ncnc2[nH]nc(Br)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 4/20 0.43
LRRK2 Q5S007 3/20 0.34
SCN9A Q15858 1/20 0.34
JAK3 P52333 2/20 0.33
FFAR2 O15552 1/20 0.33
BRAF P15056 1/20 0.32
KCNH2 Q12809 2/20 0.32
HRH3 Q9Y5N1 2/20 0.32
CA1 P00915 3/20 0.32
CA2 P00918 3/20 0.32
CA7 P43166 2/20 0.32
CA13 Q8N1Q1 2/20 0.32
ROCK2 O75116 2/20 0.31
ROCK1 Q13464 2/20 0.31
CDC42BPA Q5VT25 2/20 0.31
CDC42BPB Q9Y5S2 2/20 0.31
CA12 O43570 1/20 0.31
CA9 Q16790 1/20 0.31
NUAK1 O60285 1/20 0.30
STK16 O75716 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9980493 0.86 TNNI3K (0.36) TNNI3KLRRK2FFAR2BRAFCA1
SCHEMBL9980436 0.83 TNNI3K (0.37) TNNI3KJAK3BRAFCA1CA2
SCHEMBL9980424 0.83 TNNI3K (0.35) TNNI3KLRRK2FFAR2BRAFCA1
SCHEMBL12065601 0.77 TNNI3K (0.69) TNNI3KBRAF
SCHEMBL2226488 0.77 TNNI3K (0.47) TNNI3KLRRK2SCN9AJAK3KCNH2
SCHEMBL9980375 0.72 TNNI3K (0.40) TNNI3KBRAFCA1CA2CA7
SCHEMBL9980486 0.67 FFAR2 (0.33) LRRK2FFAR2CA1CA2CA7
SCHEMBL9980404 0.67 STK4 (0.39) TNNI3KLRRK2BRAFNUAK1STK16
SCHEMBL9980393 0.66 TNNI3K (0.40) TNNI3KBRAFCA1CA2ROCK1
SCHEMBL9980396 0.66 TNNI3K (0.44) TNNI3KBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO claimed
WO-2011149827-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC (US) 2011-12-01 WO disclosed