SCHEMBL22280595

SCHEMBL22280595

COC(=O)c1cccc(-c2cnc(Cl)o2)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.45
SLC6A4 P31645 2/20 0.42
SLC6A3 Q01959 2/20 0.42
ALDH1A1 P00352 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KDM4E B2RXH2 2/20 0.41
NPC1 O15118 2/20 0.41
HPGD P15428 2/20 0.41
RAB9A P51151 2/20 0.41
MAPT P10636 2/20 0.41
TP53 P04637 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KMT2A Q03164 3/20 0.40
HSD17B10 Q99714 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
TOP2A P11388 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22280423 0.85 FAAH (0.43) FAAHSLC6A4SLC6A3ALDH1A1SMN1; SMN2
SCHEMBL19923176 0.77 SLC6A3 (0.59) SLC6A4SLC6A3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL22280594 0.76 EDNRA (0.45) SLC6A4SLC6A3PDK2
SCHEMBL30956571 0.73 SLC6A4 (0.41) SLC6A4SLC6A3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL30956592 0.73 MRGPRX4 (0.41) SLC6A4SLC6A3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL30956550 0.72 SLC6A4 (0.40) SLC6A4SLC6A3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL30956563 0.72 KMO (0.48) SLC6A4SLC6A3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL1401560 0.72 TSHR (0.57) SLC6A4SLC6A3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL19484320 0.71 FAAH (0.55) FAAHSLC6A4SLC6A3ALDH1A1SMN1; SMN2
SCHEMBL13824070 0.71 SLC6A3 (0.53) SLC6A4SLC6A3ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020153431-A1 ESTER COMPOUND 第一三共株式会社 2020-07-30 WO disclosed
WO-2020153431-A1 ESTER COMPOUND 第一三共株式会社 2020-07-30 WO disclosed