SCHEMBL22289643

SCHEMBL22289643

CN(C(=O)CNC(=O)O)c1ccc(C#N)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.54
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
PPIB P23284 2/20 0.42
PGR P06401 4/20 0.41
RORC P51449 3/20 0.41
SIGMAR1 Q99720 2/20 0.40
TMEM97 Q5BJF2 1/20 0.40
HCRTR2 O43614 1/20 0.39
PDK2 Q15119 1/20 0.39
CACNA1G O43497 1/20 0.38
CACNA1H O95180 1/20 0.38
CACNA1I Q9P0X4 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MLNR O43193 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22289634 0.83 KMT2A (0.47) KMT2APPIBALDH1A1
SCHEMBL22312050 0.81 KMT2A (0.48) KMT2ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL22289651 0.80 FOLH1 (0.46) KMT2APPIB
SCHEMBL6170106 0.79 KMT2A (0.54) KMT2ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL22312043 0.78 KMT2A (0.52) KMT2ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL22289627 0.77 PPIB (0.61) KMT2APPIBPDK2ALDH1A1
Hydrochloric Acid SCHEMBL29472307 0.76 KMT2A (0.51) KMT2ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL1115030 0.75 PGR (0.54) KMT2ACHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL20941576 0.75 ALDH1A1 (0.51) KMT2ARORCALDH1A1
SCHEMBL1114974 0.75 PGR (0.54) KMT2ACHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3917627-A1 ACETAMIDO DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS Ideaya Biosciences, Inc. (US) 2021-12-08 EP disclosed
WO-2020160134-A1 ACETAMIDO DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2020-08-06 WO disclosed