SCHEMBL2229499

SCHEMBL2229499

CC(=O)C(C)Cc1cccc(N)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 4/20 0.45
MAOA P21397 2/20 0.43
MAOB P27338 2/20 0.43
ALDH1A1 P00352 1/20 0.42
CYP19A1 P11511 1/20 0.42
HSD11B1 P28845 1/20 0.42
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
DDX3X O00571 1/20 0.41
SLC7A5 Q01650 3/20 0.40
PNMT P11086 1/20 0.40
GRIA2 P42262 1/20 0.39
PLA2G10 O15496 1/20 0.39
PLA2G2A P14555 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28662062 0.86 ADRB2 (0.45) ADRB2MAOAMAOBALDH1A1CYP19A1
SCHEMBL1067198 0.86 PLA2G10 (0.50) ADRB2MAOAMAOBNOS3NOS1
SCHEMBL20041146 0.83 NOS1 (0.47) ALDH1A1NOS3NOS1NOS2SLC7A5
SCHEMBL23643229 0.83 NOS1 (0.47) ALDH1A1NOS3NOS1NOS2SLC7A5
SCHEMBL28133621 0.83 ADRB2 (0.45) ADRB2MAOAMAOBALDH1A1CYP19A1
SCHEMBL18500970 0.82 SLC7A5 (0.42) NOS3NOS1NOS2SLC7A5
SCHEMBL28497180 0.82 SLC7A5 (0.47) ADRB2ALDH1A1DDX3XSLC7A5
SCHEMBL28497181 0.82 SLC7A5 (0.47) ADRB2ALDH1A1DDX3XSLC7A5
SCHEMBL27744395 0.81 SMN1; SMN2 (0.43) ADRB2MAOAALDH1A1
SCHEMBL24899382 0.81 MAOB (0.45) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-55162770-A None JP disclosed
EP-2519235-A1 HETEROARYL COMPOUNDS AND USES THEREOF Avila Therapeutics, Inc. (US) 2012-11-07 EP disclosed
EP-2361248-A1 HETEROARYL COMPOUNDS AND USES THEREOF Avila Therapeutics, Inc. (US) 2011-08-31 EP disclosed
WO-2011090760-A1 HETEROARYL COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS, INC. (US) 2011-07-28 WO disclosed
WO-2009158571-A1 HETEROARYL COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS AND USES THEREOF (US) 2009-12-30 WO disclosed
JP-S55162770-A IMPROVED PREPARATION OF 2,3,3-TRIMETHYL-INDOLENINE CHISSO CORP 1980-12-18 JP disclosed