SCHEMBL18500970

SCHEMBL18500970

CC(=O)C(C)Cc1cccc(CC(C)C)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB2 P47870 1/20 0.42
PTGS1 P23219 3/20 0.41
PTGS2 P35354 3/20 0.41
LMNA P02545 2/20 0.41
CYP2C9 P11712 2/20 0.41
AKR1C3 P42330 2/20 0.41
CXCR1 P25024 2/20 0.41
CXCR2 P25025 2/20 0.41
TSHR P16473 2/20 0.41
ALB P02768 1/20 0.41
ESR1 P03372 1/20 0.41
ALOX5 P09917 1/20 0.41
RARB P10826 1/20 0.41
ADRB3 P13945 1/20 0.41
NFKB1 P19838 1/20 0.41
HTR2A P28223 1/20 0.41
NR1I3 Q14994 1/20 0.41
SLC22A6 Q4U2R8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23643229 0.86 NOS1 (0.47) SLC7A5NFKB1NOS3NOS1NOS2
SCHEMBL20041146 0.86 NOS1 (0.47) SLC7A5NFKB1NOS3NOS1NOS2
SCHEMBL18402873 0.84 SLC7A5 (0.39) SLC7A5TSHRALOX5HPGDNOS3
SCHEMBL23643117 0.84 NOS1 (0.47) SLC7A5TSHRNOS1CYP3A4
SCHEMBL9631293 0.84 MAOB (0.45) LMNA
SCHEMBL24899382 0.84 MAOB (0.45) LMNA
SCHEMBL17211514 0.84 GRIA2 (0.50) NFKB1CYP3A4
SCHEMBL2229499 0.82 ADRB2 (0.45) SLC7A5NOS3NOS1NOS2
SCHEMBL21896511 0.82 PNMT (0.61) TSHR
SCHEMBL21417673 0.82 PNMT (0.61) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9566290-B2 Boron-containing small molecules ANACOR PHARMACEUTICALS, INC. (US) 2017-02-14 US disclosed