SCHEMBL2229804

SCHEMBL2229804

CC1=CC(=O)N(c2ccccc2N2C(=O)C=CC2=O)C1=O

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 2/20 0.63
MGLL Q99685 15/20 0.58
FAAH O00519 4/20 0.49
HSP90AA1 P07900 2/20 0.41
PKM P14618 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CCR6 P51684 1/20 0.41
ATM Q13315 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TSHR P16473 1/20 0.36
RGS12 O14924 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7193393 0.92 TLR9 (0.48) TLR9MGLLFAAHPKMNPSR1
SCHEMBL2230828 0.89 MGLL (0.50) TLR9MGLLFAAHHSP90AA1PKM
SCHEMBL4846646 0.88 MGLL (0.49) TLR9MGLLFAAHHSP90AA1PKM
SCHEMBL4845238 0.88 MGLL (0.49) TLR9MGLLFAAHHSP90AA1PKM
SCHEMBL9492119 0.83 MGLL (0.60) MGLLNPSR1ALDH1A1TDP1TSHR
SCHEMBL30473083 0.83 MGLL (0.60) MGLLNPSR1ALDH1A1TDP1TSHR
SCHEMBL3679861 0.81 MGLL (0.38) TLR9MGLLFAAHHSP90AA1PKM
SCHEMBL2229875 0.80 MGLL (0.43) TLR9MGLLFAAHHSP90AA1PKM
SCHEMBL19439527 0.80 MGLL (0.56) TLR9MGLLPKMNPSR1ALDH1A1
SCHEMBL20261770 0.80 MGLL (0.59) TLR9MGLLPKMTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11230636-B2 Rubber composition having improved properties in the raw state and in the cooked state COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-01-25 US claimed
EP-3582977-B1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE MICHELIN & CIE (FR) 2021-03-31 EP claimed
US-20200056017-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2020-02-20 US claimed
WO-2018150136-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2018-08-23 WO claimed
JP-4717814-B2 2011-07-06 JP claimed
US-7442733-B2 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2008-10-28 US claimed
US-20060247342-A1 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. 2006-11-02 US claimed
EP-1664180-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE Société de Technologie Michelin (FR) 2006-06-07 EP claimed
WO-2005026250-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2005-03-24 WO claimed
US-11230636-B2 Rubber composition having improved properties in the raw state and in the cooked state COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-01-25 US disclosed
EP-3582977-B1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE MICHELIN & CIE (FR) 2021-03-31 EP disclosed
US-20200056017-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2020-02-20 US disclosed
WO-2018150136-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2018-08-23 WO disclosed
US-7442733-B2 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2008-10-28 US disclosed
US-20060247342-A1 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. 2006-11-02 US disclosed
EP-1664180-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE Société de Technologie Michelin (FR) 2006-06-07 EP disclosed
WO-2005026250-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2005-03-24 WO disclosed