SCHEMBL2230828

SCHEMBL2230828

CC1=CC(=O)N(c2cccc(N3C(=O)C=CC3=O)c2C)C1=O

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 15/20 0.50
TLR9 Q9NR96 2/20 0.48
FAAH O00519 2/20 0.42
HSP90AA1 P07900 2/20 0.40
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
CCR6 P51684 1/20 0.36
ATM Q13315 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
XPO1 O14980 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3679861 0.93 MGLL (0.38) MGLLTLR9FAAHHSP90AA1ALDH1A1
SCHEMBL2229804 0.89 TLR9 (0.63) MGLLTLR9FAAHHSP90AA1ALDH1A1
SCHEMBL4846646 0.88 MGLL (0.49) MGLLTLR9FAAHHSP90AA1ALDH1A1
SCHEMBL144793 0.85 MGLL (0.65) MGLLTLR9FAAHHSP90AA1ALDH1A1
SCHEMBL4845238 0.81 MGLL (0.49) MGLLTLR9FAAHHSP90AA1ALDH1A1
SCHEMBL7193393 0.81 TLR9 (0.48) MGLLTLR9FAAHPKMNPSR1
SCHEMBL28480530 0.80 MGLL (0.37) MGLLTLR9FAAHHSP90AA1ALDH1A1
SCHEMBL8886650 0.80 POLB (0.42) MGLLTLR9ALDH1A1PKMNPSR1
SCHEMBL2229875 0.77 MGLL (0.43) MGLLTLR9FAAHHSP90AA1ALDH1A1
SCHEMBL9492119 0.77 MGLL (0.60) MGLLALDH1A1NPSR1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11230636-B2 Rubber composition having improved properties in the raw state and in the cooked state COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-01-25 US claimed
EP-3582977-B1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE MICHELIN & CIE (FR) 2021-03-31 EP claimed
US-20200056017-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2020-02-20 US claimed
WO-2018150136-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2018-08-23 WO claimed
JP-4717814-B2 2011-07-06 JP claimed
US-7442733-B2 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2008-10-28 US claimed
US-20060247342-A1 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. 2006-11-02 US claimed
EP-1664180-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE Société de Technologie Michelin (FR) 2006-06-07 EP claimed
WO-2005026250-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2005-03-24 WO claimed
US-11230636-B2 Rubber composition having improved properties in the raw state and in the cooked state COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-01-25 US disclosed
EP-3582977-B1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE MICHELIN & CIE (FR) 2021-03-31 EP disclosed
US-20200056017-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2020-02-20 US disclosed
WO-2018150136-A1 RUBBER COMPOSITION HAVING IMPROVED PROPERTIES IN THE RAW STATE AND IN THE COOKED STATE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2018-08-23 WO disclosed
US-7442733-B2 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. (CH) 2008-10-28 US disclosed
US-20060247342-A1 Rubber composition comprising a citraconimidomaleimide MICHELIN RECHERCHE ET TECHNIQUE S.A. 2006-11-02 US disclosed
EP-1664180-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE Société de Technologie Michelin (FR) 2006-06-07 EP disclosed
WO-2005026250-A1 RUBBER COMPOSITION COMPRISING A CITRACONIMIDO-MALEIMIDE SOCIETE DE TECHNOLOGIE MICHELIN (FR) 2005-03-24 WO disclosed