SCHEMBL2229840

SCHEMBL2229840

Oc1ccccc1Nc1nncs1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.49
P2RY1 P47900 1/20 0.46
ALOX5 P09917 1/20 0.46
TAAR1 Q96RJ0 1/20 0.45
MIF P14174 1/20 0.45
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 3/20 0.43
HPGD P15428 2/20 0.43
TSHR P16473 2/20 0.42
CYP1A2 P05177 3/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA5A P35218 1/20 0.41
CA5B Q9Y2D0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213060 0.72 MAPK1 (0.53) MAPTP2RY1TAAR1ALDH1A1KDM4E
SCHEMBL31069449 0.71 ALDH1A1 (0.59) ALOX5ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL8528008 0.71 MAPT (0.46) MAPTALOX5ALDH1A1KDM4EHPGD
SCHEMBL304891 0.71 CXCR2 (0.54) MAPTALDH1A1KDM4EHPGDPOLB
SCHEMBL16904081 0.70 AMY1A (0.49) MAPTALOX5TAAR1MIFALDH1A1
SCHEMBL1920752 0.69 CXCR2 (0.52) MAPTALDH1A1KDM4EHPGDPOLB
SCHEMBL3587772 0.68 MAPT (0.53) MAPTTAAR1MIFALDH1A1KDM4E
SCHEMBL15688032 0.68 MECP2 (0.51) MAPTP2RY1POLBMEN1GAA
SCHEMBL6374941 0.67 MAPT (0.47) MAPTP2RY1TAAR1MIFALDH1A1
SCHEMBL5959497 0.66 GBA1 (0.51) MAPTALDH1A1KDM4ETSHRCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2343287-A1 New 2-aminothiadiazole derivatives Almirall, S.A. (ES) 2011-07-13 EP disclosed