SCHEMBL2229994

SCHEMBL2229994

CCCCNS(=O)(=O)c1ccccc1Br

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.88
CA12 O43570 3/20 0.61
CA9 Q16790 3/20 0.61
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
CYP2C19 P33261 2/20 0.50
TSHR P16473 2/20 0.50
MEN1 O00255 1/20 0.50
TP53 P04637 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
POLB P06746 1/20 0.50
ALDH1A1 P00352 2/20 0.48
CCR1 P32246 1/20 0.46
PLCG1 P19174 1/20 0.46
FABP4 P15090 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA4 P22748 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21089221 0.90 RECQL (0.77) RECQLCA12CA9KMT2ATDP1
SCHEMBL3723910 0.83 RECQL (0.63) RECQLCA12CA9CYP1A2CYP3A4
SCHEMBL15915838 0.83 RECQL (0.68) RECQLCA12CA9CYP1A2CYP3A4
SCHEMBL4529161 0.82 RECQL (0.66) RECQLCA12CA9POLBALDH1A1
SCHEMBL12571016 0.82 RECQL (0.70) RECQLCA12CA9CYP1A2CYP3A4
SCHEMBL9577146 0.81 RECQL (0.78) RECQLCA12CA9CYP1A2CYP3A4
SCHEMBL9577217 0.81 RECQL (0.78) RECQLCA12CA9CYP1A2CYP3A4
SCHEMBL10455162 0.81 RECQL (0.78) RECQLCA12CA9CYP1A2CYP3A4
SCHEMBL9577137 0.81 RECQL (0.78) RECQLCA12CA9CYP1A2CYP3A4
SCHEMBL9462811 0.81 CA12 (0.63) RECQLCA12CA9CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091407-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLP (US) 2011-07-28 WO disclosed
WO-2011090929-A1 DUAL-ACTING THIOPHENE, PYRROLE, THIAZOLE AND FURAN ANTIHYPERTENSIVE AGENTS THERAVANCE, INC. (US) 2011-07-28 WO disclosed
WO-2003101381-A2 1,2 DIAMIDO CYCLOALKYL SODIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2003-12-11 WO disclosed