SCHEMBL22307703

SCHEMBL22307703

CCOC(=O)c1cc(C)c2[nH]c(-c3cccc(Br)c3C)nc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 5/20 0.43
PKN1 Q16512 1/20 0.40
PKN2 Q16513 1/20 0.40
PTGES O14684 1/20 0.39
ALOX5 P09917 1/20 0.39
SIRT1 Q96EB6 4/20 0.39
SIRT3 Q9NTG7 2/20 0.39
RAB9A P51151 5/20 0.38
NPC1 O15118 4/20 0.38
MAPT P10636 3/20 0.38
CYP1A2 P05177 1/20 0.36
S1PR1 P21453 1/20 0.36
PARP1 P09874 1/20 0.36
KDM4E B2RXH2 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
HCRTR1 O43613 2/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31521803 0.80 MMP2 (0.39) RAB9ANPC1MAPTKDM4ESMN1; SMN2
SCHEMBL22307190 0.80 MMP2 (0.39) RAB9ANPC1MAPTKDM4ESMN1; SMN2
SCHEMBL29473086 0.80 MMP2 (0.39) RAB9ANPC1MAPTKDM4ESMN1; SMN2
SCHEMBL22308214 0.78 HPGD (0.36) PTGESRAB9ANPC1CYP1A2S1PR1
SCHEMBL22307226 0.77 CDK9 (0.36) RAB9ANPC1MAPTCYP1A2KDM4E
SCHEMBL29473228 0.77 CDK9 (0.36) RAB9ANPC1MAPTCYP1A2KDM4E
SCHEMBL29473070 0.71 HPGD (0.34) RAB9ANPC1CYP1A2S1PR1SMN1; SMN2
SCHEMBL22307222 0.71 HPGD (0.34) RAB9ANPC1CYP1A2S1PR1SMN1; SMN2
SCHEMBL3707021 0.71 CA12 (0.42) SIRT2PKN1PKN2SIRT1SIRT3
SCHEMBL13830587 0.70 TP53 (0.50) RAB9ANPC1MAPTSMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020156323-A1 IMMUNOMODULATORS, COMPOSITIONS AND METHODS THEREOF BETTA PHARMACEUTICALS CO., LTD (CN) 2020-08-06 WO disclosed