SCHEMBL22309141

SCHEMBL22309141

O=C1CNC(c2ccc(OCC3CC3)c(C(F)(F)F)c2)=NN1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
XDH P47989 1/20 0.43
PDE3B Q13370 6/20 0.42
PDE3A Q14432 6/20 0.42
CTSS P25774 6/20 0.41
CTSK P43235 1/20 0.41
SYK P43405 2/20 0.40
TRPA1 O75762 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
AAK1 Q2M2I8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22308838 0.96 HPGD (0.42) HPGDXDHPDE3BPDE3ACTSS
SCHEMBL22307805 0.85 PDE3B (0.40) XDHPDE3BPDE3ACTSSCTSK
SCHEMBL22307809 0.85 PDE3B (0.40) XDHPDE3BPDE3ACTSSCTSK
SCHEMBL22307810 0.84 CTSS (0.46) PDE3BPDE3ACTSSCTSK
SCHEMBL22307799 0.83 PDE3B (0.55) XDHPDE3BPDE3ACTSSCTSK
SCHEMBL22309158 0.83 PDE3B (0.56) PDE3BPDE3ACTSSCTSKAAK1
SCHEMBL22307812 0.83 PDE3B (0.50) PDE3BPDE3ACTSSCTSKAAK1
SCHEMBL22309142 0.83 XDH (0.49) XDHPDE3BPDE3AAAK1
SCHEMBL22309147 0.82 S1PR1 (0.46) PDE3BPDE3ACTSSSYKHTR2C
SCHEMBL22309160 0.81 PDE3B (0.40) PDE3BPDE3ACTSSCTSKSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020157189-A1 1,2,4-TRIAZIN-6(1H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed