SCHEMBL22309147

SCHEMBL22309147

O=C1CNC(c2ccc(OCc3ccccc3)c(C(F)(F)F)c2)=NN1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.46
CTSS P25774 1/20 0.46
S1PR4 O95977 1/20 0.41
S1PR3 Q99500 1/20 0.41
S1PR5 Q9H228 1/20 0.41
MRGPRX4 Q96LA9 6/20 0.40
RXRA P19793 2/20 0.40
RXRB P28702 2/20 0.40
RXRG P48443 2/20 0.40
PDE3B Q13370 2/20 0.39
PDE3A Q14432 2/20 0.39
PTPN1 P18031 1/20 0.39
HTT P42858 1/20 0.38
SYK P43405 1/20 0.38
HTR2C P28335 1/20 0.38
SLC6A4 P31645 1/20 0.38
HTR2B P41595 1/20 0.38
PTGER1 P34995 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22307810 0.84 CTSS (0.46) S1PR1CTSSPDE3BPDE3A
SCHEMBL22309158 0.83 PDE3B (0.56) S1PR1CTSSS1PR4S1PR5RXRA
SCHEMBL22307799 0.83 PDE3B (0.55) S1PR1CTSSPDE3BPDE3A
SCHEMBL22308858 0.82 PDE3B (0.45) S1PR1CTSSMRGPRX4PDE3BPDE3A
SCHEMBL22308346 0.82 PDE3B (0.40) S1PR1CTSSRXRARXRBRXRG
SCHEMBL22309141 0.82 HPGD (0.46) CTSSPDE3BPDE3ASYKHTR2C
SCHEMBL22307812 0.82 PDE3B (0.50) S1PR1CTSSS1PR4S1PR5RXRA
SCHEMBL22309142 0.82 XDH (0.49) PDE3BPDE3A
SCHEMBL22309148 0.81 AAK1 (0.44) PDE3BPDE3A
SCHEMBL22308819 0.80 PDE3B (0.47) RXRARXRBRXRGPDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020157189-A1 1,2,4-TRIAZIN-6(1H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed