SCHEMBL22309168

SCHEMBL22309168

O=C1CNC(c2ccc(-c3ccncc3)c(C(F)(F)F)c2)=NN1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 19/20 0.53
PDE3A Q14432 19/20 0.53
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22308361 0.90 PDE3B (0.56) PDE3BPDE3A
SCHEMBL22308893 0.85 PDE3B (0.50) PDE3BPDE3A
SCHEMBL22308356 0.85 PDE3B (0.57) PDE3BPDE3AS1PR1S1PR3
SCHEMBL22308851 0.82 PDE3B (0.54) PDE3BPDE3A
SCHEMBL22309155 0.82 PDE3B (0.47) PDE3BPDE3A
SCHEMBL22308343 0.81 PDE3B (0.39) PDE3BPDE3A
SCHEMBL22308344 0.81 PDE3B (0.41) PDE3BPDE3A
SCHEMBL22307817 0.79 PDE3B (0.62) PDE3BPDE3A
SCHEMBL7355155 0.78 KCNH2 (0.44) PDE3BPDE3A
SCHEMBL22309166 0.77 PDE3B (0.54) PDE3BPDE3AS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020157189-A1 1,2,4-TRIAZIN-6(1H)-ONE COMPOUNDS FOR THE TREATMENT OF HYPERPROLIFERATIVE DISEASES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-06 WO disclosed