SCHEMBL22309751

SCHEMBL22309751

Oc1ccn2c(n1)nc1cc(Br)ccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
RAD51 Q06609 2/20 0.33
BACE1 P56817 1/20 0.33
LCK P06239 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
PABPC1 P11940 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22309752 0.87 NPM1 (0.37) MAPTNPC1ALDH1A1MAPK1RAB9A
SCHEMBL18548700 0.79 MCL1 (0.39) ALDH1A1ALOX15TSHRSMN1; SMN2MCL1
SCHEMBL29660262 0.79 MCL1 (0.39) ALDH1A1ALOX15TSHRSMN1; SMN2MCL1
SCHEMBL22309750 0.77 TP53 (0.36) MAPTNPC1ALDH1A1TP53ALOX15
SCHEMBL2163722 0.76 PTPN1 (0.44) MAPTNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL31031257 0.73 ALDH1A1 (0.41) MAPTNPC1ALDH1A1TP53ALOX15
SCHEMBL29660237 0.72 ALDH1A1 (0.49) MAPTNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL18548712 0.72 ALDH1A1 (0.49) MAPTNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL22310380 0.69 NPM1 (0.35) MAPTALOX15BACE1CYP1A2CYP2C19
SCHEMBL19714775 0.68 ALDH1A1 (0.45) MAPTNPC1ALDH1A1TP53ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3919492-A1 PYRIMIDINYL GROUP-CONTAINING TRICYCLIC COMPOUND SERVING AS C-MET INHIBITOR Medshine Discovery Inc. (CN) 2021-12-08 EP disclosed
WO-2020156453-A1 PYRIMIDINYL GROUP-CONTAINING TRICYCLIC COMPOUND SERVING AS C-MET INHIBITOR 南京明德新药研发有限公司 2020-08-06 WO disclosed