SCHEMBL2231791

SCHEMBL2231791

CCCC/C(=C\C(=O)O)c1cc(C)c(Oc2ccc(OCc3ccc(OC(F)F)cc3)cn2)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 7/20 0.40
ALKBH1 Q13686 1/20 0.38
PSEN1 P49768 11/20 0.37
ALOX5 P09917 8/20 0.37
PTGES O14684 6/20 0.37
ACACB O00763 4/20 0.36
MRGPRX4 Q96LA9 1/20 0.35
ACACA Q13085 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2231793 0.86 PPARG (0.48) PPARGPSEN1ALOX5PTGES
SCHEMBL2235842 0.84 TDP1 (0.37) PPARGALKBH1PSEN1ALOX5PTGES
SCHEMBL2233200 0.84 ALOX5 (0.35) PPARGALOX5ACACBMRGPRX4ACACA
SCHEMBL2232578 0.83 PDPK1 (0.34) MRGPRX4
SCHEMBL13581943 0.81 ALKBH1 (0.40) ALKBH1ACACBMRGPRX4ACACA
SCHEMBL13581942 0.81 ALKBH1 (0.40) ALKBH1ACACBMRGPRX4ACACA
SCHEMBL2231788 0.80 APP (0.38) PPARGALKBH1PTGESACACB
SCHEMBL2234688 0.78 MAOB (0.41) ACACBMRGPRX4ACACA
SCHEMBL2234682 0.78 MAOB (0.41) ACACBMRGPRX4ACACA
SCHEMBL2234686 0.78 MAOB (0.41) ACACBMRGPRX4ACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011093524-A1 DI - SUBSTITUTED PYRIDINE DERIVATIVES AS ANTICANCERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2011-08-04 WO disclosed