SCHEMBL22322698

SCHEMBL22322698

O=c1[nH]c(Br)cc2cc(Br)ccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 2/20 0.55
CDC25B P30305 1/20 0.55
CASP6 P55212 1/20 0.55
PPP1CA P62136 1/20 0.55
APAF1 O14727 1/20 0.47
METAP2 P50579 1/20 0.46
CHEK1 O14757 3/20 0.41
PIM1 P11309 2/20 0.41
FLT3 P36888 2/20 0.41
AURKA O14965 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
PRKD3 O94806 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
ABL1 P00519 1/20 0.41
NTRK1 P04629 1/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL392734 0.81 GAA (0.59) TDP2CDC25BCASP6PPP1CAAPAF1
SCHEMBL1818129 0.78 KDM4E (0.60) TDP2CDC25BCASP6APAF1GAA
SCHEMBL12302517 0.77 TDP2 (0.49) TDP2CDC25BCASP6PPP1CAAPAF1
SCHEMBL24801287 0.77 TDP2 (0.49) TDP2CDC25BCASP6PPP1CAAPAF1
SCHEMBL26126207 0.72 CDC25B (1.00) TDP2CDC25BCASP6PPP1CAAPAF1
SCHEMBL14927075 0.72 KDM4E (0.41) GAAMAPTNPSR1TYMSHPGD
SCHEMBL7588 0.72 AHR (0.53) TDP2CDC25BCASP6PPP1CAMETAP2
SCHEMBL21812417 0.70 CYP19A1 (0.55) METAP2CHEK1PIM1FLT3AURKA
SCHEMBL29735151 0.69 METAP2 (0.56) TDP2CDC25BCASP6PPP1CAAPAF1
SCHEMBL396016 0.69 METAP2 (0.56) TDP2CDC25BCASP6PPP1CAAPAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115572262-A Isoquinoline derivative and preparation method thereof 厦门沃克沃德医药科技有限公司 2023-01-06 CN disclosed
EP-3920922-A1 DIHYDROOROTATE DEHYDROGENASE INHIBITORS Janssen Biotech, Inc. (US) 2021-12-15 EP disclosed
WO-2020161663-A1 DIHYDROOROTATE DEHYDROGENASE INHIBITORS JANSSEN BIOTECH, INC. (US) 2020-08-13 WO disclosed