SCHEMBL2234414

SCHEMBL2234414

CC(C)(C)N(C(=O)O)[C@H]1CN(Cc2ccccc2)c2ccccc2NC1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 1/20 0.49
EPHX2 P34913 1/20 0.48
BRD4 O60885 3/20 0.42
CACNA1G O43497 3/20 0.42
CACNA1H O95180 3/20 0.42
CACNA1I Q9P0X4 3/20 0.42
HDAC2 Q92769 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
HDAC6 Q9UBN7 4/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
MTNR1A P48039 2/20 0.38
MTNR1B P49286 2/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
BRS3 P32247 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2234153 0.83 KMT2A (0.37) BRD4KDM4EALDH1A1NPC1GAA
SCHEMBL2234145 0.83 KMT2A (0.37) BRD4KDM4EALDH1A1NPC1GAA
SCHEMBL14386531 0.76 ALOX12 (0.71) ALOX12EPHX2BRD4CACNA1GCACNA1H
SCHEMBL6178932 0.74 SCN9A (0.49) ALOX12EPHX2BRD4HDAC2HDAC8
SCHEMBL12345856 0.74 EPHX2 (0.59) ALOX12EPHX2BRD4CACNA1GCACNA1H
SCHEMBL12345855 0.74 SCN9A (0.49) ALOX12EPHX2BRD4HDAC2HDAC8
SCHEMBL3910690 0.74 EPHX2 (0.53) ALOX12EPHX2BRD4CACNA1GCACNA1H
SCHEMBL17312583 0.73 RIPK1 (0.39) EPHX2KDM4EALDH1A1NPC1GAA
SCHEMBL17312584 0.73 RIPK1 (0.39) EPHX2KDM4EALDH1A1NPC1GAA
Hydrochloric Acid SCHEMBL2236123 0.73 EPHX2 (0.58) ALOX12EPHX2BRD4CACNA1GCACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7994161-B2 Derivatives of 2-alkoxy-3,4,5-trihydroxy-alkyl amides, preparation and use thereof, and compositions containing the same SANOFI-AVENTIS (FR) 2011-08-09 US disclosed