SCHEMBL223517

SCHEMBL223517

CCCCc1ccc(N(c2ccc(C)cc2)c2ccc(C3C=CC(c4ccccc4)(N(c4ccc(C)cc4)c4ccc(CCCC)cc4)C=C3)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.38
HSD11B1 P28845 2/20 0.33
HRH1 P35367 3/20 0.32
OPRL1 P41146 1/20 0.32
KCNH2 Q12809 2/20 0.32
BCHE P06276 1/20 0.31
DRD3 P35462 2/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CYP2C19 P33261 1/20 0.30
CHRM2 P08172 1/20 0.30
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
CHRM1 P11229 1/20 0.30
DRD1 P21728 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
ADRA1A P35348 1/20 0.30
OPRM1 P35372 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2268708 0.91 CNR2 (0.33) CNR2HSD11B1
SCHEMBL221878 0.90 CNR2 (0.31) CNR2HSD11B1
SCHEMBL223877 0.85 HSD11B1 (0.31) HSD11B1OPRL1
SCHEMBL4213708 0.81 ALDH1A1 (0.35) CYP2C19ALDH1A1
SCHEMBL8862830 0.77
SCHEMBL10042897 0.75 CNR2 (0.55) CNR2HSD11B1KCNH2BCHEDRD3
SCHEMBL13197732 0.75 CNR2 (0.55) CNR2HSD11B1KCNH2BCHEDRD3
SCHEMBL12831536 0.75 CNR2 (0.55) CNR2HSD11B1KCNH2BCHEDRD3
SCHEMBL12313700 0.72 CA2 (0.52) CNR2KCNH2CA1CA2CHRM2
SCHEMBL4570447 0.72 CA2 (0.52) CNR2KCNH2CA1CA2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 179 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3309618-A1 POLYCARBONATE CONTAINING PHOTOCONDUCTORS Xerox Corporation (US) 2018-04-18 EP claimed
US-9851647-B1 Polycarbonate containing photoconductors XEROX CORPORATION (US) 2017-12-26 US claimed
EP-2278405-B1 Methods of making a photoreceptor outer layer XEROX CORP (US) 2017-04-19 EP claimed
EP-2293145-B1 Overcoat layer comprising core-shell fluorinated particles XEROX CORP (US) 2016-08-03 EP claimed
US-20150261105-A1 BIPHENYL POLYCARBONATE CONTAINING PHOTOCONDUCTORS XEROX CORPORATION (US) 2015-09-17 US claimed
US-9128392-B2 Polyarylatecarbonate containing photoconductors XEROX CORPORATION (US) 2015-09-08 US claimed
US-9069268-B2 Polyarylatecarbonate fluoropolymer containing photoconductors XEROX CORPORATION (US) 2015-06-30 US claimed
US-20150147690-A1 POLYARYLATECARBONATE CONTAINING PHOTOCONDUCTORS XEROX CORPORATION (US) 2015-05-28 US claimed
US-20150079511-A1 POLYARYLATECARBONATE FLUOROPOLYMER CONTAINING PHOTOCONDUCTORS XEROX CORPORATION (US) 2015-03-19 US claimed
US-20140356772-A1 TERPENE POLYCARBONATE CONTAINING PHOTOCONDUCTORS XEROX CORPORATION (US) 2014-12-04 US claimed
US-20110053064-A1 OVERCOAT LAYER COMPRISING CORE-SHELL FLUORINATED PARTICLES XEROX CORPORATION (US) 2011-03-03 US claimed
EP-2278405-A1 Methods of making an improved photoreceptor outer layer Xerox Corporation (US) 2011-01-26 EP claimed
EP-2278406-A1 Photoreceptor outer layer Xerox Corporation (US) 2011-01-26 EP claimed
US-20110014563-A1 METHODS OF MAKING AN IMPROVED PHOTORECEPTOR OUTER LAYER XEROX CORPORATION (US) 2011-01-20 US claimed
US-20110014557-A1 PHOTORECEPTOR OUTER LAYER XEROX CORPORATION (US) 2011-01-20 US claimed
US-7807324-B2 Photoconductors XEROX CORPORATION (US) 2010-10-05 US claimed
US-7718336-B2 Photoconductors containing photogenerating chelating components XEROX CORPORATION (US) 2010-05-18 US claimed
US-7662526-B2 Photoconductors XEROX CORPORATION (US) 2010-02-16 US claimed
US-20090263737-A1 IMAGING MEMBER AND METHODS OF FORMING THE SAME XEROX CORPORATION (US) 2009-10-22 US claimed
US-20080070136-A1 Photoconductors XEROX CORPORATION 2008-03-20 US claimed