SCHEMBL2235592

SCHEMBL2235592

OB(O)c1cnc(C=S)nc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA7 P43166 1/20 0.31
ENPP2 Q13822 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15120297 0.75 KDM4E (0.44) CA4CA6CA5ACA7ENPP2
SCHEMBL7452989 0.70 ENPP2 (0.39) CA4CA6CA5ACA7ENPP2
SCHEMBL2238608 0.69
SCHEMBL154802 0.69 CA2 (0.42) CA4CA6CA5ACA7ENPP2
SCHEMBL9523 0.69 HDAC1 (0.38) CA4CA6CA5ACA7ENPP2
SCHEMBL1427905 0.69 ENPP2 (0.42) CA4CA6CA5ACA7ENPP2
SCHEMBL4556016 0.69 ENPP2 (0.33) CA4CA6CA5ACA7ENPP2
SCHEMBL16361627 0.69 ENPP2 (0.33) CA4CA6CA5ACA7ENPP2
SCHEMBL21469007 0.69 HDAC8 (0.36) CA4CA6CA5ACA7ENPP2
Hydrochloric Acid SCHEMBL29955269 0.67 HDAC1 (0.37) CA4CA6CA5ACA7ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012127212-A1 IMIDAZO [1, 2 - B] PYRIDAZINE DERIVATIVES AS CDPK1 INHIBITORS MEDICAL RESEARCH COUNCIL TECHNOLOGY (GB) 2012-09-27 WO disclosed
WO-2011101640-A1 FUSED HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF MALARIA MEDICAL RESEARCH COUNCIL TECHNOLOGY (GB) 2011-08-25 WO disclosed