SCHEMBL22360323

SCHEMBL22360323

O=C(c1cnc(N2CC(CO)(CO)C2)nc1)N1CCC(N2C=Cc3ccccc3C2)CC1

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 13/20 0.41
DGAT2 Q96PD7 5/20 0.39
PDE4B Q07343 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22360365 0.87 ADRA1A (0.55) ADRA1ADGAT2
SCHEMBL22360349 0.85 ADRA1A (0.52) ADRA1ADGAT2
SCHEMBL22345196 0.81 ADRA1A (0.60) ADRA1A
SCHEMBL22360324 0.78 ADRA1A (0.46) ADRA1ADGAT2
SCHEMBL22360348 0.72 ADRA1A (0.57) ADRA1ADGAT2
SCHEMBL22345185 0.69 ADRA1A (0.60) ADRA1ADGAT2
SCHEMBL16824482 0.67 ADRA1A (0.80) ADRA1A
SCHEMBL28294761 0.67 PARP1 (0.37)
SCHEMBL22345162 0.65 POLB (0.53)
SCHEMBL22360326 0.64 ADRA1A (0.61) ADRA1ADGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020165031-A1 SUBSTITUTED ISOQUINOLINE-PIPERIDINYLMETHANONE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2020-08-20 WO disclosed