SCHEMBL2236352

SCHEMBL2236352

CC(C)CCC(=O)Nc1cccc(B2OC(C)(C)C(C)(C)O2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
NAMPT P43490 1/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
LIPG Q9Y5X9 2/20 0.40
AAK1 Q2M2I8 2/20 0.40
LPL P06858 1/20 0.40
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12350692 0.84 NAMPT (0.37) NAMPTKDM4EMAPTNPC1RAB9A
SCHEMBL3264202 0.83 GAA (0.56) CA1CA2CA9MAPTNPC1
SCHEMBL1851971 0.83 MAP4K4 (0.43) CA1CA2CA9KDM4ERAB9A
SCHEMBL18343188 0.82 ALDH1A1 (0.47) CA1CA2CA9KDM4EMAPT
SCHEMBL28663994 0.81 SMN1; SMN2 (0.50) CA1CA2CA9KDM4EMAPT
SCHEMBL17078435 0.80 PTPRC (0.50) L3MBTL1HDAC3HDAC4HDAC1HDAC7
SCHEMBL2236402 0.80 LMNA (0.50) CA1CA2CA9MAPTSMN1; SMN2
SCHEMBL19801178 0.79 CA1 (0.39) CA1CA2CA9LIPGAAK1
SCHEMBL16150246 0.79 HSD17B10 (0.52) CA1CA2CA9KDM4EHSD17B10
SCHEMBL2357751 0.79 ALDH1A1 (0.54) KDM4EMAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101640-A1 FUSED HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF MALARIA MEDICAL RESEARCH COUNCIL TECHNOLOGY (GB) 2011-08-25 WO disclosed