SCHEMBL2236450

SCHEMBL2236450

NC(CC(=O)O)NC(=O)c1cccnc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.53
ECE1 P42892 1/20 0.53
HDAC1 Q13547 2/20 0.53
HDAC6 Q9UBN7 1/20 0.53
THRB P10828 1/20 0.53
EPHX2 P34913 3/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
PLOD2 O00469 1/20 0.50
CYP3A4 P08684 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HIF1A Q16665 1/20 0.49
ALDH1A1 P00352 1/20 0.49
APP P05067 1/20 0.49
GAA P10253 1/20 0.49
HCAR3 P49019 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471469 0.86 HDAC1 (0.58) LMNAECE1HDAC1HDAC6THRB
SCHEMBL2234114 0.82 SLC1A2 (0.54) LMNAHDAC1HDAC6NPC1RAB9A
SCHEMBL27739096 0.82 CASP3 (0.60) LMNAECE1HDAC1HDAC6THRB
SCHEMBL14660540 0.82 CASP3 (0.60) LMNAECE1HDAC1HDAC6THRB
SCHEMBL30038032 0.82 CASP3 (0.60) LMNAECE1HDAC1HDAC6THRB
SCHEMBL2240935 0.81 CYP1A2 (0.55) EPHX2CYP2C9CYP2C19PLOD2CYP3A4
SCHEMBL16031690 0.81 LMNA (0.55) LMNAECE1HDAC1HDAC6THRB
SCHEMBL27868838 0.78 LMNA (0.52) LMNAECE1HDAC1HDAC6THRB
SCHEMBL30037941 0.77 CA2 (0.54) LMNAECE1HDAC1HDAC6THRB
SCHEMBL28830880 0.77 CA2 (0.54) LMNAECE1HDAC1HDAC6THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2531520-A1 TEMPLATE-FIXED PEPTIDOMIMETICS WITH CXCR7 MODULATING ACTIVITY Polyphor AG (CH) 2012-12-12 EP disclosed
WO-2011095607-A1 TEMPLATE-FIXED PEPTIDOMIMETICS WITH CXCR7 MODULATING ACTIVITY POLYPHOR AG (CH) 2011-08-11 WO disclosed