SCHEMBL22368668

SCHEMBL22368668

CC1CC(=O)CC2CCC2c2cccc(Br)c2C1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
BRD4 O60885 1/20 0.32
KDM4E B2RXH2 1/20 0.32
KDM1A O60341 1/20 0.31
PDE7A Q13946 1/20 0.31
MAP1LC3B Q9GZQ8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23053830 0.68 KDM1A (0.42) ALDH1A1BRD4KDM4EKDM1A
SCHEMBL7936463 0.67 BRD4 (0.39) BRD4PDE7A
SCHEMBL1699423 0.66 PIM1 (0.43) ALDH1A1MAPK1SMN1; SMN2BRD4KDM4E
SCHEMBL30422252 0.66 BRD4 (0.39) BRD4
SCHEMBL13360866 0.66 BRD4 (0.39) BRD4
SCHEMBL19518238 0.63 CREBBP (0.61) ALDH1A1BRD4
SCHEMBL16315955 0.63 CYP1A2 (0.33) HTTKDM4E
SCHEMBL15773405 0.62 HSD11B1 (0.48)
SCHEMBL2968862 0.61 ALDH1A1 (0.38) ALDH1A1CYP3A4CYP2D6CYP2C9LMNA
SCHEMBL1073565 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3204360-B1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH INC (US) 2020-08-26 EP disclosed