SCHEMBL22369248

SCHEMBL22369248

COC(=O)N1CCC(C)C(C)(O)C1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.39
USP2 O75604 2/20 0.38
TSHR P16473 3/20 0.37
CYP2C9 P11712 5/20 0.37
CYP1A2 P05177 4/20 0.37
CYP2D6 P10635 4/20 0.37
ALDH1A1 P00352 1/20 0.37
CHRNB2 P17787 2/20 0.37
CHRNA4 P43681 2/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CYP3A4 P08684 4/20 0.35
CYP2C19 P33261 3/20 0.35
HSD17B10 Q99714 2/20 0.35
BRD4 O60885 2/20 0.35
BRDT Q58F21 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20312244 0.80 CYP2C9 (0.40) EPHX1USP2TSHRCYP2C9CYP1A2
SCHEMBL13709104 0.76 EPHX1 (0.33) EPHX1USP2CYP2C9CYP1A2CYP2D6
SCHEMBL12883924 0.74 EPHX1 (0.38) EPHX1USP2TSHRCYP2C9CYP1A2
SCHEMBL23714589 0.74 EPHX1 (0.41) EPHX1USP2TSHRCYP2C9CYP1A2
SCHEMBL12883927 0.74 HSD11B1 (0.41) EPHX1TSHRCYP2C9ALDH1A1
SCHEMBL20312912 0.74 CYP2D6 (0.35) EPHX1USP2TSHRCYP2C9CYP1A2
SCHEMBL771850 0.72 GAA (0.53) EPHX1TSHRALDH1A1CHRNB2CHRNA4
SCHEMBL31597078 0.72 EPHX1 (0.38) EPHX1USP2TSHRCYP2C9CYP1A2
SCHEMBL24606819 0.71 CYP1A2 (0.47) USP2TSHRCYP2C9CYP1A2CYP2D6
SCHEMBL17176084 0.71 USP2 (0.51) USP2TSHRCYP2C9CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3313844-B1 HETEROARYL SUBSTITUTED AMINOPYRIDINE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2020-08-26 EP disclosed