SCHEMBL2238908

SCHEMBL2238908

CS(=O)(=O)n1cc(CCNc2cc(-c3cccnc3)ncn2)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 15/20 0.51
CYP3A4 P08684 15/20 0.51
CLK4 Q9HAZ1 12/20 0.51
HSD17B10 Q99714 11/20 0.51
CYP2C19 P33261 10/20 0.51
CYP2D6 P10635 9/20 0.51
ALDH1A1 P00352 8/20 0.51
ALOX15 P16050 5/20 0.51
USP2 O75604 2/20 0.51
TSHR P16473 2/20 0.49
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
KDM4E B2RXH2 3/20 0.46
HPGD P15428 2/20 0.46
HTR6 P50406 2/20 0.44
IDE P14735 1/20 0.42
NR1D1 P20393 1/20 0.40
TP53 P04637 2/20 0.39
MAPK1 P28482 2/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2242579 0.85 HTR6 (0.41) CYP1A2CYP3A4CLK4HSD17B10CYP2C19
SCHEMBL2239882 0.72 PTGDR (0.42) CYP1A2CYP3A4CLK4HSD17B10CYP2C19
SCHEMBL11992443 0.70 HTR6 (0.73) HTR6IDE
SCHEMBL19355276 0.69 CYP1A2 (0.52) CYP1A2CYP3A4CLK4HSD17B10CYP2C19
SCHEMBL10820371 0.66 HTR6 (0.71) HTR6
SCHEMBL20816293 0.66 CYP1A2 (0.62) CYP1A2CYP3A4CLK4HSD17B10CYP2C19
SCHEMBL19355422 0.64 CYP1A2 (0.46) CYP1A2CYP3A4CLK4HSD17B10CYP2C19
SCHEMBL2244628 0.64 CYP1A2 (0.59) CYP1A2CYP3A4CLK4HSD17B10CYP2C19
SCHEMBL9056570 0.63 HTR2C (0.51) HSD17B10MEN1KMT2AKDM4EHPGD
SCHEMBL7671291 0.63 HTR6 (0.66) HTR6IDE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989458-B2 Pyrimidine derivatives as alk-5 inhibitors NOVARTIS AG (CH) 2011-08-02 US claimed