SCHEMBL22396

SCHEMBL22396

Cc1cc(-c2csc(C(=O)c3cccc(O)c3)c2)ccc1O

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 20/20 0.69
HSD17B2 P37059 20/20 0.69
CYP3A4 P08684 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C19 P33261 1/20 0.59
HSD17B14 Q9BPX1 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22898 0.81 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C19
SCHEMBL31415 0.77 HSD17B1 (0.65) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C19
SCHEMBL10353029 0.76 HSD17B1 (0.79) HSD17B1HSD17B2HSD17B14
SCHEMBL1180208 0.74 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C19
SCHEMBL23296 0.73 HSD17B1 (0.48) HSD17B1HSD17B2
SCHEMBL29848168 0.72 HSD17B1 (0.96) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C19
SCHEMBL12656410 0.72 HSD17B1 (0.96) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C19
SCHEMBL30431 0.72 HSD17B1 (1.00) HSD17B1HSD17B2
SCHEMBL31061230 0.70 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2D6CYP2C19
SCHEMBL9390168 0.70 HSD17B1 (0.51) HSD17B1HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO claimed
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed