SCHEMBL23296

SCHEMBL23296

COc1cccc(C(=O)c2cc(-c3ccc(OC)c(C)c3)cs2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.48
HSD17B2 P37059 3/20 0.48
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
CYP2C8 P10632 1/20 0.43
PARP1 P09874 1/20 0.42
STS P08842 2/20 0.41
NPC1 O15118 3/20 0.41
HPGD P15428 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
PGR P06401 1/20 0.40
AR P10275 1/20 0.40
ABL1 P00519 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23735 0.81 HSD17B2 (0.60) HSD17B1HSD17B2
SCHEMBL30916784 0.79 TUBB4A (0.58) HSD17B1HSD17B2MAPTMEN1KMT2A
SCHEMBL23127 0.76 CES2 (0.54) CES2CES1CYP2C8PARP1STS
SCHEMBL30916762 0.75 TUBB4A (0.45) L3MBTL1
SCHEMBL22396 0.73 HSD17B1 (0.69) HSD17B1HSD17B2
SCHEMBL23360 0.72 HSD17B1 (0.64) HSD17B1HSD17B2
SCHEMBL30916805 0.72 TUBB4A (0.61) ALDH1A1MAPTL3MBTL1
SCHEMBL23339 0.71 HSD17B2 (0.66) HSD17B1HSD17B2MAPK13MAPK12MAPK11
SCHEMBL30916744 0.71 MAPT (0.53) HPGDALDH1A1MAPTKDM4ECNR2
SCHEMBL6870004 0.71 HSD17B1 (0.64) HSD17B1HSD17B2PARP1NPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed