SCHEMBL22397495

SCHEMBL22397495

O=C(O)N1CC=Cc2ncccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 2/20 0.36
KDM4E B2RXH2 4/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 5/20 0.33
ALDH1A1 P00352 2/20 0.33
TSHR P16473 2/20 0.33
MAPT P10636 2/20 0.33
CYP3A4 P08684 1/20 0.33
ALOX15 P16050 1/20 0.33
BLM P54132 1/20 0.33
AGER Q15109 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NAPRT Q6XQN6 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
LMNA P02545 2/20 0.32
TP53 P04637 1/20 0.32
GAA P10253 1/20 0.32
KDM6B O15054 1/20 0.31
KDM6A O15550 1/20 0.31
TET3 O43151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27770600 0.89 L3MBTL1 (0.34) MYCKDM4ETDP1L3MBTL1ALDH1A1
SCHEMBL16671338 0.86 PARP1 (0.36) MYCKDM4ETSHRNAPRTSMN1; SMN2
SCHEMBL28984504 0.79 POLB (0.43) POLB
SCHEMBL27857904 0.76 GAA (0.32) MYCGAA
Quinoline SCHEMBL28157604 0.75 ALDH1A1 (0.44) KDM4EALDH1A1MAPTCYP3A4ALOX15
SCHEMBL12671549 0.74 SMN1; SMN2 (0.33) MYCKDM4EALDH1A1MAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL27458213 0.73 GAA (0.30) GAA
SCHEMBL29376182 0.73 P2RX4 (0.44) TSHRNPSR1SMN1; SMN2LMNAKMT2A
SCHEMBL27303243 0.72 TRIM24 (0.30)
SCHEMBL27779336 0.72 GRIA2 (0.31) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3703692-A1 NOVEL SUBSTITUTED TETRAHYDROQUINOLIN COMPOUNDS AS INDOLEAMINE 2,3-DIOXYGENASE (IDO) INHIBITORS Merck Sharp & Dohme Corp. (US) 2020-09-09 EP disclosed