SCHEMBL22447435

SCHEMBL22447435

Cc1cnc(C)c(NS(=O)(=O)c2sc(C)nc2C)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.43
ITK Q08881 1/20 0.39
SLC40A1 Q9NP59 6/20 0.39
PIK3CG P48736 1/20 0.36
PIK3CA P42336 3/20 0.36
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
BRAF P15056 1/20 0.35
LMNA P02545 3/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
NPY5R Q15761 1/20 0.34
HSD11B1 P28845 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22447427 0.86 KIT (0.42) KITITKPIK3CGPIK3CAPIK3CD
SCHEMBL22508613 0.84 KIT (0.40) KITITKPIK3CGPIK3CAPIK3CD
SCHEMBL22447413 0.78 ALPL (0.39) KITITKPIK3CAHSD11B1
SCHEMBL25389991 0.73 PIK3CA (0.46) KITPIK3CGPIK3CAPIK3CDPIK3CB
SCHEMBL31185557 0.73 PIK3CA (0.46) KITPIK3CGPIK3CAPIK3CDPIK3CB
SCHEMBL24576532 0.73 PIK3C3 (0.48) PIK3CGPIK3CAPIK3CDPIK3CBHTT
SCHEMBL12459761 0.72 THRB (0.51) KITPIK3CABRAFLMNAPKM
SCHEMBL18595669 0.70 BRD4 (0.44) PIK3CGPIK3CALMNAALDH1A1SMN1; SMN2
SCHEMBL22447465 0.69 SLC22A12 (0.44) KITITKPIK3CGPIK3CAPIK3CD
SCHEMBL925786 0.69 PIK3CB (0.50) PIK3CGPIK3CAPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3712143-A1 QUINAZOLINONE COMPOUND AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2020-09-23 EP disclosed