SCHEMBL22448601

SCHEMBL22448601

CC(C)c1cnc(Br)cc1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 6/20 0.45
GABRB1 P18505 4/20 0.45
LMNA P02545 3/20 0.42
SLC6A2 P23975 2/20 0.42
HTR2B P41595 2/20 0.42
TRPA1 O75762 1/20 0.42
CHRM1 P11229 1/20 0.42
ADRA1A P35348 1/20 0.42
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
GABRB2 P47870 4/20 0.38
HSP90AA1 P07900 6/20 0.34
HSP90AB1 P08238 5/20 0.34
HPGD P15428 2/20 0.33
FAAH O00519 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
GABRG2 P18507 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23749845 0.79 GABRA1 (0.39) GABRA1GABRB1CA1CA2GABRB2
SCHEMBL15614474 0.76 GABRA1 (0.37) GABRA1GABRB1LMNASLC6A2HTR2B
SCHEMBL25613928 0.76 GABRA1 (0.37) GABRA1GABRB1CA1CA2
SCHEMBL12197721 0.76 SLC6A2 (0.48) GABRA1GABRB1LMNASLC6A2HTR2B
SCHEMBL22448790 0.75 LMNA (0.44) GABRA1GABRB1LMNASLC6A2HTR2B
SCHEMBL22448704 0.74 LMNA (0.42) GABRA1GABRB1LMNASLC6A2HTR2B
SCHEMBL22448616 0.74 POLB (0.36) GABRA1GABRB1KMT2A
SCHEMBL25927987 0.74 GABRA1 (0.35) GABRA1GABRB1LMNA
SCHEMBL23510746 0.74 LMNA (0.42) GABRA1GABRB1LMNASLC6A2HTR2B
SCHEMBL16248167 0.74 LMNA (0.48) GABRA1GABRB1LMNASLC6A2HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3964505-A1 SOLID FORM OF DIAMINOPYRIMIDINE COMPOUND OR HYDRATE THEREOF, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF Beijing Tide Pharmaceutical Co., Ltd. (CN) 2022-03-09 EP disclosed
EP-3712144-A1 P2X3 AND/OR P2X2/3 RECEPTOR ANTAGONIST, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF Beijing Tide Pharmaceutical Co., Ltd. (CN) 2020-09-23 EP disclosed