SCHEMBL22448616

SCHEMBL22448616

CC(C)c1cnc(Br)cc1N

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
UHRF1 Q96T88 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
P2RX3 P56373 9/20 0.35
P2RX2 Q9UBL9 9/20 0.35
DHFR P00374 1/20 0.32
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23749845 0.79 GABRA1 (0.39) GABRA1GABRB1P2RX3P2RX2
SCHEMBL26064376 0.77 NOS3 (0.44) POLBGAAGFERUHRF1GABRA1
SCHEMBL25841159 0.76 NOS3 (0.38) POLBGAAGFERUHRF1P2RX3
SCHEMBL25613928 0.76 GABRA1 (0.37) GABRA1GABRB1P2RX3P2RX2
SCHEMBL15614474 0.76 GABRA1 (0.37) POLBGAAGFERUHRF1GABRA1
SCHEMBL25843328 0.76 UHRF1 (0.52) POLBGAAGFERUHRF1P2RX3
SCHEMBL22448726 0.75 POLB (0.42) POLBGAAGFERP2RX3P2RX2
SCHEMBL22448601 0.74 GABRA1 (0.45) GABRA1GABRB1KMT2A
SCHEMBL12132818 0.74 P2RX3 (0.38) POLBGAAGFERUHRF1GABRA1
SCHEMBL25927987 0.74 GABRA1 (0.35) POLBGAAGFERUHRF1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3712144-A1 P2X3 AND/OR P2X2/3 RECEPTOR ANTAGONIST, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF Beijing Tide Pharmaceutical Co., Ltd. (CN) 2020-09-23 EP disclosed