SCHEMBL22448701

SCHEMBL22448701

CC(C)c1cnc(Br)cc1OCC#N

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.33
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
ALOX15 P16050 1/20 0.31
HTT P42858 1/20 0.31
ALOX5AP P20292 2/20 0.31
FEN1 P39748 2/20 0.31
P2RX3 P56373 2/20 0.31
P2RX2 Q9UBL9 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22448793 0.83 POLB (0.36) POLBALDH1A1GAAALOX15HTT
SCHEMBL22448669 0.78 JAK2 (0.34) POLBALDH1A1GAAALOX15HTT
SCHEMBL22448805 0.77 POLB (0.32) POLBALDH1A1GAAALOX15HTT
SCHEMBL5529615 0.76 LMNA (0.45) POLBALDH1A1GAAGABRA1GABRB1
SCHEMBL22448705 0.75 POLB (0.46) POLBGAAP2RX3P2RX2
SCHEMBL1494087 0.75 P2RX3 (0.47) P2RX3P2RX2
SCHEMBL19364184 0.73 P2RX3 (0.42) POLBALDH1A1GAAP2RX3P2RX2
SCHEMBL22448614 0.73 KMT2A (0.33) ALDH1A1GAAGABRA1GABRB1ALOX15
SCHEMBL25484238 0.72 ALDH1A1 (0.50) ALDH1A1
SCHEMBL22448625 0.72 MAPK1 (0.47) ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3964505-A1 SOLID FORM OF DIAMINOPYRIMIDINE COMPOUND OR HYDRATE THEREOF, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF Beijing Tide Pharmaceutical Co., Ltd. (CN) 2022-03-09 EP disclosed
EP-3712144-A1 P2X3 AND/OR P2X2/3 RECEPTOR ANTAGONIST, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF Beijing Tide Pharmaceutical Co., Ltd. (CN) 2020-09-23 EP disclosed