SCHEMBL224499

SCHEMBL224499

BrC1=COc2ccccc2C1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
OXTR P30559 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
CYP1A2 P05177 1/20 0.31
GAA P10253 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
AHR P35869 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL295062 0.76 MAOA (0.50) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL2013569 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL295061 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL30714851 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL4551344 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL18280613 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL276642 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL1707855 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL230114 0.71 ESR2 (0.50) MAOAMAOBOXTRABCG2GAA
SCHEMBL5541287 0.69 MAOA (0.43) MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115724834-A Indenoquinolinone or chromene quinolinone derivative and preparation method and application thereof 广东工业大学 2023-03-03 CN claimed
CN-115724834-B Indenoquinolinone or chromenequinolinone derivative as well as preparation method and application thereof 广东工业大学 2025-03-21 CN disclosed
CN-115724834-A Indenoquinolinone or chromene quinolinone derivative and preparation method and application thereof 广东工业大学 2023-03-03 CN disclosed
EP-1577288-B1 Selective estrogen receptor modulators EISAI R&D MAN CO LTD (JP) 2014-07-23 EP disclosed
US-8399520-B2 Selective estrogen receptor modulator EISAI R&D MANAGEMENT CO., LTD. (JP) 2013-03-19 US disclosed
US-20120004315-A1 Selective Estrogen Receptor Modulator RADIUS HEALTH, INC. 2012-01-05 US disclosed
US-7960412-B2 Selective estrogen receptor modulator EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-06-14 US disclosed
US-20090325930-A1 SELECTIVE ESTROGEN RECEPTOR MODULATOR RADIUS HEALTH, INC. 2009-12-31 US disclosed
US-7612114-B2 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-11-03 US disclosed
US-20060116364-A1 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI CO., LTD. (JP) 2006-06-01 US disclosed
EP-1577288-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS Eisai Co., Ltd. (JP) 2005-09-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325930-A1 SELECTIVE ESTROGEN RECEPTOR MODULATOR ESR1, GPER1, ESR2 MAOA 3273/4885MAOB 3449/4885OXTR 151/4885
US-20060116364-A1 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer BRCA1, BCR, RCC1 MAOA 4367/4885MAOB 4319/4885OXTR 843/4885
US-20120004315-A1 Selective Estrogen Receptor Modulator ESR1, GPER1, ESR2 MAOA 3358/4885MAOB 3399/4885OXTR 110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.