SCHEMBL1707855

SCHEMBL1707855

OC1=COc2ccccc2C1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.48
MAOB P27338 2/20 0.48
ESR2 Q92731 1/20 0.37
OXTR P30559 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
ITGB2 P05107 1/20 0.32
ICAM1 P05362 1/20 0.32
ITGAL P20701 1/20 0.32
CYP1A2 P05177 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
GAA P10253 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30
DRD4 P21917 1/20 0.30
DRD5 P21918 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30714851 1.00 MAOA (0.48) MAOAMAOBESR2OXTRABCG2
SCHEMBL295062 0.76 MAOA (0.50) MAOAMAOBESR2OXTRABCG2
SCHEMBL18280613 0.74 MAOA (0.48) MAOAMAOBESR2OXTRABCG2
SCHEMBL295061 0.74 MAOA (0.48) MAOAMAOBESR2OXTRABCG2
SCHEMBL2013569 0.74 MAOA (0.48) MAOAMAOBESR2OXTRABCG2
SCHEMBL4551344 0.74 MAOA (0.48) MAOAMAOBESR2OXTRABCG2
SCHEMBL276642 0.74 MAOA (0.48) MAOAMAOBOXTRABCG2ITGB2
SCHEMBL224499 0.74 MAOA (0.48) MAOAMAOBESR2OXTRABCG2
SCHEMBL7977979 0.74 MAOA (0.43) MAOAMAOBESR2
SCHEMBL16397646 0.72 MAOA (0.42) MAOAMAOBOXTRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111423405-A Method for synthesizing benzopyran 3 alcohol derivative compound 浙江工业大学 2020-07-17 CN claimed
JP-3575767-B2 2004-10-13 JP claimed
EP-0764157-A1 BENZOPYRANS AND THEIR USE AS THERAPEUTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-03-26 EP claimed
WO-1995034545-A1 BENZOPYRANS AND THEIR USE AS THERAPEUTIC AGENTS SMITHKLINE BEECHAM PLC (GB) 1995-12-21 WO claimed
EP-0677519-A1 CHROMAN DERIVATIVE AND MEDICINAL USE THEREOF Japan Tobacco Inc. (JP) 1995-10-18 EP claimed
EP-0673373-A1 BICYCLIC COMPOUNDS WITH PHARMACEUTICAL ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-09-27 EP claimed
EP-0413438-A1 Benzopyran compounds Beecham Group p.l.c. (GB) 1991-02-20 EP claimed
WO-2026088071-A1 SUBSTITUTED FUSED HETEROARYL LACTAM COMPOUNDS PFIZER INC. (US) 2026-04-30 WO disclosed
CN-111423405-B Method for synthesizing benzopyran 3 alcohol derivative compound 浙江工业大学 2021-11-26 CN disclosed
CN-111423405-A Method for synthesizing benzopyran 3 alcohol derivative compound 浙江工业大学 2020-07-17 CN disclosed
US-20140088030-A1 WATER SOLUBLE AND ACTIVABLE PHENOLICS DERIVATIVES WITH DERMOCOSMETIC AND THERAPEUTIC APPLICATIONS AND PROCESS FOR PREPARING SAID DERIVATIVES LIBRAGEN (FR) 2014-03-27 US disclosed
EP-2027279-B1 Phenolic compounds with cosmetic and therapeutic applications LIBRAGEN (FR) 2012-04-18 EP disclosed
US-20110183930-A1 WATER SOLUBLE AND ACTIVABLE PHENOLICS DERIVATIVES WITH DERMOCOSMETIC AND THERAPEUTIC APPLICATIONS AND PROCESS FOR PREPARING SAID DERIVATIVES LIBRAGEN (FR) 2011-07-28 US disclosed
EP-0547523-A1 Ethanolates of 6-sulfonylsubstituted 3-hydroxychromanes and their use as inhalation means for illnesses HOECHST AKTIENGESELLSCHAFT (DE) 1993-06-23 EP disclosed
WO-1993005045-A1 SPIROCYCLIC BENZOPYRAN IMIDAZOLINES THE UPJOHN COMPANY (US) 1993-03-18 WO disclosed
EP-0516658-A1 BENZOPYRANS HAVING PHARMACOLOGICAL ACTIVITY BEECHAM GROUP PLC (GB) 1992-12-09 EP disclosed
WO-1991011446-A1 BENZOPYRANS HAVING PHARMACOLOGICAL ACTIVITY BEECHAM GROUP PLC (GB) 1991-08-08 WO disclosed
EP-0412760-A2 Benzopyran derivatives Beecham Group p.l.c. (GB) 1991-02-13 EP disclosed
EP-0373204-A1 NOVEL COMPOUNDS AND TREATMENT BEECHAM GROUP PLC (GB) 1990-06-20 EP disclosed
WO-1989010925-A1 NOVEL COMPOUNDS AND TREATMENT BEECHAM GROUP PLC (GB) 1989-11-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110183930-A1 WATER SOLUBLE AND ACTIVABLE PHENOLICS DERIVATIVES WITH DERMOCOSMETIC AND THERAPEUTIC APPLICATIONS AND PROCESS FOR PREPARING SAID DERIVATIVES UGGT1, TYR, G6PD MAOA 688/4885MAOB 981/4885ESR2 2662/4885
US-20140088030-A1 WATER SOLUBLE AND ACTIVABLE PHENOLICS DERIVATIVES WITH DERMOCOSMETIC AND THERAPEUTIC APPLICATIONS AND PROCESS FOR PREPARING SAID DERIVATIVES UGGT1, TYR, G6PD MAOA 688/4885MAOB 981/4885ESR2 2662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.