SCHEMBL2245261

SCHEMBL2245261

COc1cccc(COc2ccc(-c3ccc(C(=O)N[C@@H](CCC(=O)O)C(N)=O)cc3)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.56
HPGDS O60760 3/20 0.53
DHFR P00374 2/20 0.50
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
KMT2A Q03164 1/20 0.48
PTPN1 P18031 1/20 0.47
FFAR1 O14842 6/20 0.47
MAOB P27338 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB2 P47870 1/20 0.46
AKR1B1 P15121 1/20 0.46
FFAR4 Q5NUL3 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2250713 0.96 MMP12 (0.54) MMP12HPGDSDHFRKDM4ENPC1
SCHEMBL2243988 0.91 MMP12 (0.53) MMP12HPGDSDHFRALDH1A1POLB
SCHEMBL2247647 0.90 MMP12 (0.62) MMP12HPGDSDHFRPTPN1FFAR1
SCHEMBL2245262 0.89 MRGPRX4 (0.53) DHFRKDM4ENPC1ALDH1A1LMNA
SCHEMBL2251669 0.88 MMP12 (0.61) MMP12HPGDSDHFRALDH1A1PTPN1
SCHEMBL2246953 0.88 GRM5 (0.57) MMP12HPGDSDHFRPTPN1MAOB
SCHEMBL2247420 0.88 MMP12 (0.56) MMP12HPGDSDHFRNPC1ALDH1A1
SCHEMBL3583723 0.87 KLKB1 (0.54) DHFRNPC1RAB9A
SCHEMBL2250678 0.87 MMP12 (0.54) MMP12HPGDSALDH1A1POLBGAA
SCHEMBL2250715 0.85 MRGPRX4 (0.51) DHFRKDM4ENPC1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed