SCHEMBL2247647

SCHEMBL2247647

NC(=O)[C@H](CCC(=O)O)NC(=O)c1ccc(-c2ccc(OCc3cccc(-c4ccccc4)c3)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.62
HPGDS O60760 5/20 0.59
FFAR1 O14842 6/20 0.57
AKR1B1 P15121 1/20 0.57
FFAR4 Q5NUL3 1/20 0.57
NR1H4 Q96RI1 1/20 0.55
DHFR P00374 2/20 0.53
PTPN1 P18031 1/20 0.52
PTGER4 P35408 1/20 0.49
PTGER3 P43115 1/20 0.49
F2 P00734 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2251669 0.94 MMP12 (0.61) MMP12HPGDSFFAR1DHFRPTPN1
SCHEMBL2250713 0.93 MMP12 (0.54) MMP12HPGDSFFAR1AKR1B1FFAR4
SCHEMBL2246953 0.91 GRM5 (0.57) MMP12HPGDSDHFRPTPN1
SCHEMBL2247420 0.91 MMP12 (0.56) MMP12HPGDSFFAR1AKR1B1FFAR4
SCHEMBL2245261 0.90 MMP12 (0.56) MMP12HPGDSFFAR1AKR1B1FFAR4
SCHEMBL2248588 0.90 MMP12 (0.57) MMP12HPGDSFFAR1AKR1B1FFAR4
SCHEMBL2247651 0.88 MRGPRX4 (0.56) HPGDSFFAR1AKR1B1FFAR4NR1H4
SCHEMBL3577147 0.87 KLKB1 (0.56) FFAR1AKR1B1FFAR4NR1H4DHFR
SCHEMBL2252391 0.85 MMP12 (0.66) MMP12HPGDSPTPN1
SCHEMBL2243988 0.85 MMP12 (0.53) MMP12HPGDSDHFRPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed