SCHEMBL2245262

SCHEMBL2245262

COc1cccc(COc2ccc(-c3ccc(C(=O)N[C@@H](CCC(N)=O)C(=O)O)cc3)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.53
DHFR P00374 3/20 0.50
PTPN1 P18031 1/20 0.49
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
GPR132 Q9UNW8 5/20 0.48
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
KMT2A Q03164 1/20 0.48
CA2 P00918 2/20 0.47
CA1 P00915 1/20 0.47
FPGS Q05932 1/20 0.47
C3AR1 Q16581 1/20 0.46
TP53 P04637 1/20 0.46
PKM P14618 1/20 0.46
NFKB1 P19838 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2250715 0.96 MRGPRX4 (0.51) MRGPRX4DHFRPTPN1RAB9ASMN1; SMN2
SCHEMBL2243990 0.91 DHFR (0.50) MRGPRX4DHFRPTPN1ALDH1A1GPR132
SCHEMBL2247651 0.90 MRGPRX4 (0.56) MRGPRX4DHFRGPR132CA2CA1
SCHEMBL2245261 0.89 MMP12 (0.56) DHFRPTPN1RAB9ASMN1; SMN2KDM4E
SCHEMBL2251677 0.88 GPR132 (0.55) MRGPRX4DHFRPTPN1ALDH1A1GPR132
SCHEMBL2246956 0.88 GRM5 (0.57) MRGPRX4DHFRCA2CA1
SCHEMBL2247421 0.88 PARP15 (0.56) MRGPRX4DHFRRAB9ASMN1; SMN2NPC1
SCHEMBL2250684 0.87 POLB (0.46) MRGPRX4PTPN1ALDH1A1POLBGAA
SCHEMBL6030433 0.86 GPR132 (0.65) PTPN1RAB9AGPR132POLBGAA
SCHEMBL2250713 0.85 MMP12 (0.54) DHFRRAB9ASMN1; SMN2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed