SCHEMBL22452978

SCHEMBL22452978

CC(=N)c1cc(NC(=O)c2c(C)cc(N)c(N)c2C)ccc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.51
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
MAPT P10636 1/20 0.38
FADS1 O60427 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
CYP26A1 O43174 1/20 0.35
CYP26B1 Q9NR63 1/20 0.35
CYP1A2 P05177 1/20 0.34
CFTR P13569 1/20 0.34
GUSB P08236 1/20 0.34
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
PLG P00747 1/20 0.33
PLAU P00749 1/20 0.33
PLAT P00750 1/20 0.33
KLK1 P06870 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453892 0.82 LRRK2 (0.55) LRRK2NPC1RAB9AFADS1SMN1; SMN2
SCHEMBL22453804 0.78 LRRK2 (0.45) LRRK2NPC1RAB9AMAPTFADS1
SCHEMBL22890421 0.76 LRRK2 (0.48) LRRK2NPC1RAB9AMAPTFADS1
SCHEMBL22453793 0.76 LRRK2 (0.46) LRRK2NPC1RAB9AMAPTFADS1
SCHEMBL22452996 0.75 LRRK2 (0.50) LRRK2NPC1RAB9AMAPTLMNA
SCHEMBL22453875 0.74 LRRK2 (0.46) LRRK2NPC1RAB9AMAPTFADS1
SCHEMBL22453384 0.74 LRRK2 (0.50) LRRK2RAB9AFADS1SMN1; SMN2ALDH1A1
SCHEMBL22890305 0.74 LRRK2 (0.59) LRRK2FADS1ALDH1A1F2F10
SCHEMBL22452969 0.72 LRRK2 (0.48) LRRK2NPC1RAB9AFADS1SMN1; SMN2
SCHEMBL22453902 0.72 LRRK2 (0.58) LRRK2FADS1HTTF2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020191261-A1 INDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2020-09-24 WO disclosed